BDBM50469353 CHEMBL4283353

SMILES CCC[C@H](C)Nc1ncc2c(cn([C@H]3CC[C@H](O)CC3)c2n1)-c1ccc(CN2CCCN(C)CC2)cc1

InChI Key InChIKey=HYUGTGGDEAGXJP-HRNNMHKYSA-N

Data  4 KI  28 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50469353   

TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Unc Eshelman School of Pharmacy

Curated by ChEMBL

LigandBDBM50469353(CHEMBL4283353)Copy SMILESCopy InChI

Affinity DataIC50: >100nMAssay Description:Inhibition of N-terminal GST-tagged human KIT cytoplasmic domain (544 to 976 end residues) expressed in baculovirus expression system using fluorecen...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPurchasePC cidPC sid

In DepthDetails ArticlePubMed
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